產(chǎn)品屬性:
產(chǎn)品名稱 | CTAP TFA |
規(guī)格 | 1mg、5mg、10mg |
貨號(hào) | EY-01Y12198 |
Cas No.: N/A
別名: N/A
化學(xué)名: N/A
分子式: C53H70F3N13O12S2
分子量: 1218.32
溶解度: H2O: 100 mg/mL (82.08 mM)
儲(chǔ)存條件: Store at -20°C
General tipsFor obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.
Shipping ConditionEvaluation sample solution : ship with blue ice
All other available size: ship with RT , or blue ice upon request
產(chǎn)品描述:
CTAP TFA is a potent, highly selective, and brain penetrant μ opioid receptor antagonist (IC50=3.5 nM) and displays over 1200-fold selectivity over δ opioid (IC50=4500 nM) and somatostatin receptors. CTAP TFA can be used for the study of L-DOPA-induced dyskinesia (LID)[1].[1]. Mitchell J Bartlett, et al. Highly-selective μ-opioid Receptor Antagonism Does Not Block L-DOPA-induced Dyskinesia in a Rodent Model.BMC Res Notes
特別提醒公司產(chǎn)品僅供科研使用